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ANALYSIS OF EZH2 MUTATIONS IN SOLID AND LIQUID BIOPSY AND ITS ROLE AS PREDICTIVE MARKER FOR CHEMOTHERAPY IN PATIENTS WITH FOLLICULAR LYMPHOMA
Author(s): ,
Laura Sanz-Villanueva
Affiliations:
Gregorio Marañón Health Research Institute (IiSGM),Madrid,Spain;Department of Hematology,Gregorio Marañón General University Hospital,Madrid,Spain
,
Francisco Díaz Crespo
Affiliations:
Pathology Department,Gregorio Marañón General University Hospital,Madrid,Spain
,
Reyes Martín Rojas
Affiliations:
Department of Hematology,Gregorio Marañón General University Hospital,Madrid,Spain
,
Diego Carbonell
Affiliations:
Gregorio Marañón Health Research Institute (IiSGM),Madrid,Spain;Department of Hematology,Gregorio Marañón General University Hospital,Madrid,Spain
,
María Chicano
Affiliations:
Gregorio Marañón Health Research Institute (IiSGM),Madrid,Spain;Department of Hematology,Gregorio Marañón General University Hospital,Madrid,Spain
,
Julia Suárez-González
Affiliations:
Gregorio Marañón Health Research Institute (IiSGM),Madrid,Spain;Genomics Unit,Gregorio Marañón General University Hospital,Madrid,Spain
,
Paula Muñiz
Affiliations:
Gregorio Marañón Health Research Institute (IiSGM),Madrid,Spain;Department of Hematology,Gregorio Marañón General University Hospital,Madrid,Spain
,
Javier Menarguez
Affiliations:
Department of Hematology,Gregorio Marañón General University Hospital,Madrid,Spain;Pathology Department,Gregorio Marañón General University Hospital,Madrid,Spain
,
Mi Kwon
Affiliations:
Gregorio Marañón Health Research Institute (IiSGM),Madrid,Spain;Department of Hematology,Gregorio Marañón General University Hospital,Madrid,Spain
,
Jose Luis Diez Martín
Affiliations:
Gregorio Marañón Health Research Institute (IiSGM),Madrid,Spain;Department of Hematology,Gregorio Marañón General University Hospital,Madrid,Spain;Department of Medicine,School of Medicine, Complutense University of Madrid,Madrid,Spain
,
Ismael Buño
Affiliations:
Gregorio Marañón Health Research Institute (IiSGM),Madrid,Spain;Department of Hematology,Gregorio Marañón General University Hospital,Madrid,Spain;Genomics Unit,Gregorio Marañón General University Hospital,Madrid,Spain;Department of Cellular Biology,School of Medicine, Complutense University of Madrid,Madrid,Spain
,
Carolina Martínez-Laperche
Affiliations:
Gregorio Marañón Health Research Institute (IiSGM),Madrid,Spain;Department of Hematology,Gregorio Marañón General University Hospital,Madrid,Spain
Mariana Bastos Oreiro
Affiliations:
Gregorio Marañón Health Research Institute (IiSGM),Madrid,Spain;Department of Hematology,Gregorio Marañón General University Hospital,Madrid,Spain
EHA Library. Oreiro M. 06/09/21; 325628; EP870
Dr. Mariana Bastos Oreiro
Dr. Mariana Bastos Oreiro
Contributions
Abstract
Presentation during EHA2021: All e-poster presentations will be made available as of Friday, June 11, 2021 (09:00 CEST) and will be accessible for on-demand viewing until August 15, 2021 on the Virtual Congress platform.

Abstract: EP870

Type: E-Poster Presentation

Session title: Lymphoma Biology & Translational Research

Background

EZH2 encodes the catalytic subunit of Polycomb repressor complex (PCR2) and mediates methylation of Lys27 residue of histone H3 (H3K27). Missense mutations in EZH2 lead to decreased transcriptional function of genes involved in cell cycle regulation and plasma cell differentiation, which contributes to oncogenic transformation. EZH2 have been detected to be mutated in near 20% of follicular lymphomas (FL) and this gene is included in the risk model m7-FL International Prognostic Index (m7-FLIPI). Furthermore, EZH2 inhibitors appear as a new treatment option in FL.

Aims

We aimed to analyse retrospectively the frequency of mutations in EZH2 at diagnosis in tissue and circulating cell free DNA (cfDNA) in patients with FL and assess the patient's response to therapy, depending on the EZH2 mutation status.

Methods

We included 179 consecutive patients diagnosed with FL from 2002 to 2019. Thirty-seven patients were excluded due to insufficient DNA quantity or quality. Of the 142 analysed patients, 49 had cfDNA sample at diagnosis. DNA was extracted from solid biopsies using Maxwell(R) 16 FFPE Plus LEV DNA Purification Kit (Promega). We obtained cfDNA from plasma samples, using QIAamp® Circulating Nucleic Acid (Qiagen). RT-qPCR reactions were performed in ctDNA using PrimeTime Mini LNA probe for EZH2 Y646. Sanger sequencing were used in tumor DNA for detection of mutations in exon 16 (Y646) and 18 (A682 and A692). Clinical characteristics, therapy and outcome were collected. Data analysis including descriptive statistics and Fisher’s exact test was performed using IBM SPSS Statistics 26 (IBM, USA).

Results

Of the 142 patients analysed in tissue, 41 (29%) presented mutations in EZH2. These mutations were found in 46% of grade 3B FL and 27% of grades 1, 2 and 3A FL (Table 1). Y646 mutations in cfDNA were detected in 5/49 (10%) with EZH2 mutated in tumor and stage III-IV FL. Clinical and biological characteristics according to EZH2 mutation status in tumor were compared in patients with lower-grade FL (Table 1) and high grade 3B (data not shown). No statistical differences were found in lower grade-FL. Instead, patients with grade 3B and mutated EZH2 had statistically higher FLIPI risk (80% vs 0%; p=0.048). Overall survival (OS) of total cohort and according to therapy received and EZH2 mutation status were compared and there were no statistically significant differences. In terms of progression free survival (PFS), our results shown that mutated EZH2 patients treated with R-bendamustine were significantly associated with inferior PFS (p=0.013) (Figure 1a), unlike R-CHOP treated patients (p=0.15) (Figure 1b).

Conclusion

The frequency of EZH2 mutations in our total cohort is similar to previously reported. Mutations were more frequent in high grade FL patients. Low grade FL patients mutated at diagnosis, receiving R-bendamustine were associated with inferior PFS. The mutational status of these patients at diagnosis could be useful to guide treatment. In patients with stage III-IV, liquid biopsy may be used at diagnosis to guide on the selection of therapy, as EZH2 mutations are detectable in advanced stage FL.

Keyword(s): EZH2, Follicular lymphoma, Lymphoma therapy, Plasma

Presentation during EHA2021: All e-poster presentations will be made available as of Friday, June 11, 2021 (09:00 CEST) and will be accessible for on-demand viewing until August 15, 2021 on the Virtual Congress platform.

Abstract: EP870

Type: E-Poster Presentation

Session title: Lymphoma Biology & Translational Research

Background

EZH2 encodes the catalytic subunit of Polycomb repressor complex (PCR2) and mediates methylation of Lys27 residue of histone H3 (H3K27). Missense mutations in EZH2 lead to decreased transcriptional function of genes involved in cell cycle regulation and plasma cell differentiation, which contributes to oncogenic transformation. EZH2 have been detected to be mutated in near 20% of follicular lymphomas (FL) and this gene is included in the risk model m7-FL International Prognostic Index (m7-FLIPI). Furthermore, EZH2 inhibitors appear as a new treatment option in FL.

Aims

We aimed to analyse retrospectively the frequency of mutations in EZH2 at diagnosis in tissue and circulating cell free DNA (cfDNA) in patients with FL and assess the patient's response to therapy, depending on the EZH2 mutation status.

Methods

We included 179 consecutive patients diagnosed with FL from 2002 to 2019. Thirty-seven patients were excluded due to insufficient DNA quantity or quality. Of the 142 analysed patients, 49 had cfDNA sample at diagnosis. DNA was extracted from solid biopsies using Maxwell(R) 16 FFPE Plus LEV DNA Purification Kit (Promega). We obtained cfDNA from plasma samples, using QIAamp® Circulating Nucleic Acid (Qiagen). RT-qPCR reactions were performed in ctDNA using PrimeTime Mini LNA probe for EZH2 Y646. Sanger sequencing were used in tumor DNA for detection of mutations in exon 16 (Y646) and 18 (A682 and A692). Clinical characteristics, therapy and outcome were collected. Data analysis including descriptive statistics and Fisher’s exact test was performed using IBM SPSS Statistics 26 (IBM, USA).

Results

Of the 142 patients analysed in tissue, 41 (29%) presented mutations in EZH2. These mutations were found in 46% of grade 3B FL and 27% of grades 1, 2 and 3A FL (Table 1). Y646 mutations in cfDNA were detected in 5/49 (10%) with EZH2 mutated in tumor and stage III-IV FL. Clinical and biological characteristics according to EZH2 mutation status in tumor were compared in patients with lower-grade FL (Table 1) and high grade 3B (data not shown). No statistical differences were found in lower grade-FL. Instead, patients with grade 3B and mutated EZH2 had statistically higher FLIPI risk (80% vs 0%; p=0.048). Overall survival (OS) of total cohort and according to therapy received and EZH2 mutation status were compared and there were no statistically significant differences. In terms of progression free survival (PFS), our results shown that mutated EZH2 patients treated with R-bendamustine were significantly associated with inferior PFS (p=0.013) (Figure 1a), unlike R-CHOP treated patients (p=0.15) (Figure 1b).

Conclusion

The frequency of EZH2 mutations in our total cohort is similar to previously reported. Mutations were more frequent in high grade FL patients. Low grade FL patients mutated at diagnosis, receiving R-bendamustine were associated with inferior PFS. The mutational status of these patients at diagnosis could be useful to guide treatment. In patients with stage III-IV, liquid biopsy may be used at diagnosis to guide on the selection of therapy, as EZH2 mutations are detectable in advanced stage FL.

Keyword(s): EZH2, Follicular lymphoma, Lymphoma therapy, Plasma

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